产品
编 号:F200412
分子式:C33H34N4O3
分子量:534.65
产品类型
结构图
CAS No: 167355-22-8
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生物活性:
GV-150013 is a selective CCK-B receptor antagonist. GV-150013 has sleep aid effect.
体内研究:
GV-150013 (0.5 - 60μg/kg, 静脉注射, 给药一次) 在老年大鼠模型中增加快速动眼睡眠和非快速动眼睡眠.Animal Model:Old rats .
Dosage:0.5 μg/kg, 5μg/kg, 60μg/kg
Administration:Intraperitoneal injection, Once
Result:The duration of REM sleep and non-REM sleep was longer than that of control.