产品
编 号:F211807
分子式:C9H8N2O
分子量:160.17
产品类型
结构图
CAS No: 1769-24-0
联系客服
产品详情
生物活性:
2-Methylquinazolin-4-ol is a potent competitive poly(ADP-ribose) synthetase inhibitor, with a Ki of 1.1 μM. 2-Methylquinazolin-4-ol mammalian aspartate transcarbamylase (ATCase) inhibitor, with 0.20 mM.
体内研究:
2-Methylquinazolin-4-ol (0.2-1 mg; i.g.; for two days) inhibits ATCase in a dosedependent manner in vivo.Animal Model:Mice
Dosage:0.2 mg, 0.4 mg, 0.6 mg, 0.8 mg, 1 mg
Administration:Oral gavage, for two days
Result:Showed an inhibitory effect upon ATCase.
体外研究:
2-Methylquinazolin-4-ol inhibits ATCase in a concentration-dependent manner.