产品
编 号:F230749
分子式:C15H12ClFN6OS
分子量:378.81
产品类型
结构图
CAS No: 1848232-20-1
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产品详情
生物活性:
GSK2226649A (compound 2) is a novel activator of satellite cell proliferation and enhanced repair of damaged muscle.
体内研究:
The pharmacokinetic parameters of GSK2226649A(compound 2) in mice Dose(mg)routeCmax(ng/mL) Tmax(hrs) T1/2(hrs)AUC0-inf(h*ng/mL) 30oral13840.51.6172030SC17831.06.112077
体外研究:
GSK2226649A(compound 2) (0.1-10μM) 可以剂量依赖性促进肌肉干细胞增殖,可有效加速骨骼肌损伤体内小鼠模型中受损骨骼肌的修复。