产品
编 号:F280126
分子式:C16H16N4O2
分子量:296.32
产品类型
结构图
CAS No: 2229039-45-4
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生物活性:
(E/Z)-ZL0420 is a racemic compound of (Z)-ZL0420 and (E)-ZL0420 isomers. (E)-ZL0420 is a potent and selective bromodomain-containing protein 4 (BRD4) inhibitor with IC50 values of 27 nM against BRD4 BD1 and 32 nM against BRD4 BD2.