产品
编 号:F291094
分子式:C22H24ClF2NO2
分子量:407.88
产品类型
结构图
CAS No: 24677-86-9
联系客服
产品详情
生物活性:
Lenperone hydrochloride (AHR 2277) is an antipsychotic compound and a dopamine antagonist. Lenperone hydrochloride reduces gastroesophageal sphincter pressure of healthy dogs. Lenperone hydrochloride can be used for neurological disease research.
体内研究:
Lenperone hydrochloride (0.16 和 0.44mg/kg;肌内注射;一次) 降低健康犬的平均值胃食管括约肌压力 (GESP)。Lenperone hydrochloride (0.5,1.0 和 2.0 mg/kg;皮下注射) 在脑损伤大鼠中显示抗精神疾病的作用,诱导剂量依赖的镇静状态并减少双侧间质核、终纹。Animal Model:Healthy adult dogs
Dosage:0.16 and 0.44 mg/kg
Administration:Intramuscular injection; 0.16 and 0.44 mg/kg, once
Result:Effectively decreased gastroesophageal sphincter pressure (GESP) of dogs.