产品
编 号：F308114
分子式：C20H22N2S
分子量：322.47
分子式：C20H22N2S
分子量：322.47
产品类型
规格
价格
是否有货
10mM*1mL in DMSO
询价
询价
1mg
152
In-stock
5mg
528
In-stock
10mg
792
In-stock
25mg
1120
In-stock
50mg
1440
In-stock
100mg
1920
In-stock
结构图
CAS No: 29216-28-2
产品详情
生物活性：
Mequitazine is a potent, and long-acting histamine H1 antagonist.
体内研究：
Mequitazine and clemizole antagonize the effect of histamine in guinea-pig ileum competitively. Mequitazine at 107 produces a parallel shift of the dose-response curve to acetylcholine in the rat duodenum. Mequitazine at highest concentration shows anticholinergic activity. Mequitazine inhibits contractile responses to KCl, phenylephrine (PE), 5-hydroxytryptamine (5-HT), and Ca2+ in rat aorta.
体外研究：
Mequitazine is a potent H1-receptors selective antihistaminic drug widely studied and used for allergic disorders such as hay fever and urticaria. Mequitazine demonstrates significant bactericidal effects against all the tested clinical isolates including Ps. aeruginosa. Its effect against the Gram-positive isolates is more pronounced.
Mequitazine is a potent, and long-acting histamine H1 antagonist.
体内研究：
Mequitazine and clemizole antagonize the effect of histamine in guinea-pig ileum competitively. Mequitazine at 107 produces a parallel shift of the dose-response curve to acetylcholine in the rat duodenum. Mequitazine at highest concentration shows anticholinergic activity. Mequitazine inhibits contractile responses to KCl, phenylephrine (PE), 5-hydroxytryptamine (5-HT), and Ca2+ in rat aorta.
体外研究：
Mequitazine is a potent H1-receptors selective antihistaminic drug widely studied and used for allergic disorders such as hay fever and urticaria. Mequitazine demonstrates significant bactericidal effects against all the tested clinical isolates including Ps. aeruginosa. Its effect against the Gram-positive isolates is more pronounced.
产品资料
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