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编 号:F311293
分子式:C20H28O5
分子量:348.43
产品类型
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CAS No: 30220-46-3
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生物活性:
Ingenol is a PKC activator, with a Ki of 30 μM, with antitumor activity.
体外研究:
Ingenol is a PKC activator, with a Ki of 30 μM. Ingenol induces ornithine decarboxylase activity (1, 3 mM), and causes morphological changes (1 mM) in primary mouse epidermal keratinocytes. Ingenol (125 μM, 250 μM, 500 μM, 1 mM) also inhibits cell-cell communication.