产品
编 号:F363170
分子式:C24H39NO6
分子量:437.57
产品类型
结构图
CAS No: 466-26-2
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产品详情
生物活性:
Neoline (Bullatine B)) is the active ingredient of the active ingredient (PA), which can be used to cure the disease. Neoline Flow Suppression Nav1.7 Electrical Flow Control (VGSC),Improve diabetes mechanical pain sensitivity. Neoline has a list of compounds that can be used, research on its use, and the quality of its processing during processing in pain.
体内研究:
Neoline(10 mg/kg/天;皮下注射;10 天)可减轻奥沙利铂引起的周围神经病变。Neoline 抑制小鼠模型中紫杉醇或部分坐骨神经损伤引起的异常性疼痛。Neoline(1-10 mg/kg;皮下注射;单剂量)显示出抗伤害作用,并显着增加糖尿病小鼠的机械伤害感受阈值。
体外研究:
Neoline (1 μM) 显着降低 HEK293 细胞去极化诱导的 Nav1.7 VGSC 电流,IC50 为 25.8 nM。