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编 号:F041698
分子式:C19H27FO
分子量:290.42
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5mg
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10mg
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25mg
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生物活性:
Fluasterone is a potent G6PD inhibitor with a Ki of 0.51 μM. Fluasterone has anti-inflammatory, cancer preventive, and anti-diabetic effects. Fluasterone is orally active.

体内研究:
Fluasterone (0.2% and 0.3%; in diet for 39 days) 对糖尿病小鼠有抗高血糖作用。Fluasterone (200 μg/mouse; intradermal injection; once) 抑制 TPA 诱导的急性炎症和表皮增生作用。Animal Model:Male C57BL/KsJ db/db mice, diabetic model
Dosage:0.2% and 0.3%
Administration:In the diet for 39 days
Result:Markedly reduced plasma glucose levels.
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