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编 号:F394991
分子式:C22H27N3O5
分子量:413.47
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5mg
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10mg
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25mg
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50mg
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Physostigmine salicylate (Eserine salicylate) is a reversible acetylcholinesterase (AChE) inhibitor. Physostigmine salicylate crosses the blood-brain barrier and stimulates central cholinergic neurotransmission. Physostigmine salicylate can reverse memory deficits in transgenic mice with Alzheimer's disease. Physostigmine salicylate is also an antidote for anticholinergic poisoning.

体内研究:
Physostigmine salicylate (Eserine salicylate;0.03-0.3 mg/kg;sc;每日一次,持续 6 周) 改善 Tg (+) 小鼠的情境记忆和线索记忆缺陷。Animal Model:Heterozygous transgenic mice (Tg(+) mice)
Dosage:0.03, 0.1, and 0.3 mg/kg
Administration:SC; daily for 6 weeks
Result:Tended to normalize the contextual memory deficit in Tg(+) animals so that they became more similar to Tg(-) animals.
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