产品
编 号:F401410
分子式:C17H29ClN2O3
分子量:344.88
产品类型
结构图
CAS No: 5987-82-6
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产品详情
生物活性:
Oxybuprocaine hydrochloride (Benoxinate hydrochloride) reversibly blocks sodium channels and prevents propagation of painful nerve impulses in the cornea, conjunctiva, and sclera. Oxybuprocaine hydrochloride is used especially in ophthalmology and otolaryngology.
体内研究:
Oxybuprocaine hydrochloride (Benoxinate hydrochloride; 27.6, 51.7, 103.5, 413.9 μg; s.c.) provides a dose-dependent block to pinpricks in rats. Oxybuprocaine hydrochloride (27.6 μg) produces 100% of sensory/nociceptive block. Animal Model:Male Sprague-Dawley rats (203-253 g)
Dosage:27.6, 51.7, 103.5, 413.9 μg
Administration:SC
Result:Provided a dose-dependent block to pinpricks.