产品
编 号:F403314
分子式:C10H7NO3
分子量:189.17
产品类型
结构图
CAS No: 605-62-9
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产品详情
生物活性:
KAT8-IN-1 is a lysine (K) acetyltransferase 8 (KAT8) inhibitor, with IC50s of 141 μM (KAT8), 221 μM (KAT2B), 106 μM (KAT3B), respectively. KAT8 inhibits histone acetyltransferases (HATs), and could result in disease states, such as cancer or inflammatory diseases.
体外研究:
KAT8-IN-1 (compound 19) losses anti-oxidant activity (EC50>1 mM).