产品
编 号:F063154
分子式:C26H28N6O5S
分子量:536.6
产品类型
结构图
CAS No: 1188371-47-2
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产品详情
生物活性:
Valecobulin (CKD516) is a valine proagent of (S516) and a vascular disrupting agent (VDA). Valecobulin is a potent β-tubulin polymerization inhibitor with marked antitumor activity against murine and human solid tumors.
体内研究:
Valecobulin (5 mg/kg; intraperitoneal injection; administered on days 2, 6, 10, and 14; male BALB/C nu/nu mice) treatment shows markedly antitumor efficacy in various human tumor xenograft models.Animal Model:Male BALB/C nu/nu mice (5-6 weeks of age) with HCT-116 or HCT-15 cells
Dosage:5 mg/kg
Administration:Intraperitoneal injection; administered on days 2, 6, 10, and 14
Result:Had shown marked antitumor efficacy in various human tumor xenograft models.