产品
编 号：F600504
分子式：C5H14NO2P
分子量：151.14
分子式：C5H14NO2P
分子量：151.14
产品类型
规格
价格
是否有货
结构图
CAS No: 123691-29-2
产品详情
生物活性：
CGP36216 is a selective antagonist at GABA presynaptic receptor. CGP36216 binds to GABAB receptor with a Ki value of 0.3 μM. CGP36216 hydrochloride can be used for research of anxiety and trauma-related disorders.
体内研究：
Animal Model:Rats.
Dosage:20 μg/Rat.
Administration:Intra-VTA injection (ventral tegmental area).
Result:Abolishes CPP induced by intra-VTA injection of morphine.
体外研究：
CGP36216对GABA突触后受体无效，但在突触前受体上更为活跃。CGP36216 (100 μM)可以增加VTA-DA神经元自发放电的频率。
CGP36216 is a selective antagonist at GABA presynaptic receptor. CGP36216 binds to GABAB receptor with a Ki value of 0.3 μM. CGP36216 hydrochloride can be used for research of anxiety and trauma-related disorders.
体内研究：
Animal Model:Rats.
Dosage:20 μg/Rat.
Administration:Intra-VTA injection (ventral tegmental area).
Result:Abolishes CPP induced by intra-VTA injection of morphine.
体外研究：
CGP36216对GABA突触后受体无效，但在突触前受体上更为活跃。CGP36216 (100 μM)可以增加VTA-DA神经元自发放电的频率。
产品资料
Copyright©2015-2024 沪ICP备2022026524号-1
沪公网安备