产品
编 号:F745540
分子式:C20H27N2NaO5
分子量:398.43
产品类型
结构图
CAS No: 149404-21-7
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产品详情
生物活性:
Enalapril (MK-421) sodium is an angiotensin-converting enzyme (ACE) inhibitor, can be used for hypertensive diseases research.
体内研究:
Enalapril sodium (intraperitoneal injection, 0.03 mg/kg, once) reduces infarct volume due to middle cerebral artery occlusion and lower or higher doses are ineffective in Male NMRI mice.Animal Model:Male NMRI mice 20-40 g
Dosage:0.03 mg/kg
Administration:Intraperitoneal injection; once
Result:Reduced the area of middle cerebral artery infarction in mice at 0.03 mg/kg.
体外研究:
Enalapril sodium (10-20 μM) has an antiarrhythmic effect in ultrafiltered PV sleeve preparation isolated from canine hearts which can inhibit EAD and DAD-induced activity.Enalapril sodium (50 μM, 24 hours) inhibits the induction of apoptosis by patient serum only when used prior to treatment of HUVEC with Alzheimer's disease (AD) serum.Pure Enalapril sodium has better thermal stability than pure Enalapril.