产品
编 号:F754212
分子式:C20H20BrF3N6O2
分子量:513.31
产品类型
结构图
CAS No: 2640208-01-9
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产品详情
生物活性:
CDK7-IN-7 is a potent and selective CDK7 kinase inhibitor with an IC50 of <50 nM (Patent CN112661745A, compound T-01).
体外研究:
CDK7-IN-7 shows inhibitory against MDA?MB 231, MDA-MB453, OVCAR3, A2780, HCT-116, WiDr and Calu-6 cells (IC50 ranging from 12.21 to 144.9 nM).