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编 号:F756979
分子式:C19H29Cl2N3
分子量:370.36
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生物活性:
UHMCP1 dihydrochloride is a potent UHM domain splicing inhibitor with a Kd value of 79 μM. UHMCP1 dihydrochloride prevents the SF3b155/U2AF65 interaction. UHMCP1 dihydrochloride impacts cell viability and RNA splicing.

体外研究:
UHMCP1 dihydrochloride (0-100 μM; 24 h) impacts cell viability and splicing with an EC50 value of 140 μM in HEK293 cells.
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