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编 号:F099457
分子式:C18H16N2O3
分子量:308.33
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生物活性:
PHCCC(4Me) (THCCC), a PHCCC analog, is a dual mGluR2 (IC50 of 1.5 μM) negative allosteric modulator and mGluR3 (EC50 of 8.9 μM) positive allosteric modulator.

体外研究:
PHCCC(4Me) (THCCC; Compound 3) shows micromolar affinityfor mGluR2, with a Ki value of 0.6 μM.
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