产品
编 号:F124296
分子式:C24H19F4N5O
分子量:469.43
产品类型
结构图
CAS No: 1337531-89-1
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生物活性:
PERK-IN-4 is a potent and selective PERK (protein kinase R (PKR)-like endoplasmic reticulum kinase) inhibitor with an IC 50 of 0.3 nM. PERK is activated in response to a variety of endoplasmic reticulum stresses implicated in numerous disease states.