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编 号:F131069
分子式:C31H29N5O6S
分子量:599.66
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10mM*1mL in DMSO
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2mg
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5mg
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10mg
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25mg
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50mg
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100mg
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生物活性:
PI3K-IN-1 (XL-147 derivative 1) is a potent inhibitor of PI3K. PI3K-IN-1 (25 μM) blocks PI3K/Akt signaling pathways.

体外研究:
PI3K-IN-1 (25 μM) blocks PI3K/Akt signaling pathways. By using the PI3K inhibitor PI3K-IN-1, TGF-β1 induced transformation into myofibroblast is also inhibited, with relatively reduced expressions of α-SMA, Col-1 and Timp-1.
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